Explore GRPR gene products and cross-species
research data at TarMart platform. Discover comprehensive
biological information, expression tools, and therapeutic
insights for Homo sapiens (human), Cynomolgus monkeys, rodents
(mouse/rat), canines, felines, bovines, and equines. Your
premier destination for multi-species gene research solutions
Target
sublocation: Transmembrane Protein.
Gastrin-releasing peptide (GRP) regulates numerous functions of the gastrointestinal and central nervous systems, including release of gastrointestinal hormones, smooth muscle cell contraction, and epithelial cell proliferation and is a potent mitogen for neoplastic tissues. The effects of GRP are mediated through the gastrin-releasing peptide receptor. This receptor is a glycosylated, 7-transmembrane G-protein coupled receptor that activates the phospholipase C signaling pathway. The receptor is aberrantly expressed in numerous cancers such as those of the lung, colon, and prostate. An individual with autism and multiple exostoses was found to have a balanced translocation between chromosome 8 and a chromosome X breakpoint located within the gastrin-releasing peptide receptor gene. [provided by RefSeq, Jul 2008]
| Target ID |
GM-T99816
|
| Target Name |
GRPR
|
Gene Group ldentifer (Target Gene ID in Homo
species)
|
2925
|
| Gene ID |
100056400 (Equus caballus), 101096951 (Felis catus), 14829 (Mus musculus), 24938 (Rattus norvegicus) 2925 (Homo sapiens), 491754 (Canis lupus familiaris), 532784 (Bos taurus), 574339 (Macaca mulatta)
|
| Target Alternative Names |
BB2,BB2R,BRS2,GRP-R,GRP-preferring bombesin receptor,GRPR,Gastrin-releasing peptide receptor,Grpr
|
| Uniprot Accession |
P21729,P52500,P30550
|
| Protein Sub-location |
Transmembrane Protein
|
| Category |
Therapeutics Target
|
| Disease from KEGG |
Calcium signaling pathway, Neuroactive ligand-receptor interaction
|
| Gene Ensembl |
ENSECAG00000015277, ENSMUSG00000031364, ENSG00000126010, ENSCAFG00845030779, ENSBTAG00000007092, ENSMMUG00000023688
|
| Target Classification |
GPCR
|
Pre-made viral vector of GRPR cDNA Clones/ORF Plasmid
GRPR siRNA/miRNA/oligo for RNA interfence (RNAi)
| Cat No. | Product Name | GeneID | Species | Grade | Detail |
|---|
| pGMoligo2925 | Pre-made Human GRPR/BB2/BB2R siRNA oligo Duplex | 2925 | Human | In-vitro grade; in-vivo grade | Detail |
| pGMoligo24938 | Pre-made Rat Grpr siRNA oligo Duplex | 24938 | Rat | In-vitro grade; in-vivo grade | Detail |
| pGMoligo14829 | Pre-made Mouse Grpr/GRP-R siRNA oligo Duplex | 14829 | Mouse | In-vitro grade; in-vivo grade | Detail |
| pGMoligo574339 | Pre-made Cynomolgus/Rhesus macaque GRPR siRNA oligo Duplex | 574339 | Cynomolgus/Rhesus macaque | In-vitro grade; in-vivo grade | Detail |
| pGMoligo101096951 | Pre-made Cat/Feline GRPR siRNA oligo Duplex | 101096951 | Cat/Feline | In-vitro grade; in-vivo grade | Detail |
| pGMoligo491754 | Pre-made Dog/Canine GRPR siRNA oligo Duplex | 491754 | Dog/Canine | In-vitro grade; in-vivo grade | Detail |
| pGMoligo532784 | Pre-made Bovines/Cattle GRPR siRNA oligo Duplex | 532784 | Bovines/Cattle | In-vitro grade; in-vivo grade | Detail |
| pGMoligo100056400 | Pre-made Equine/Horse GRPR siRNA oligo Duplex | 100056400 | Equine/Horse | In-vitro grade; in-vivo grade | Detail |
GRPR antibody/GMab
| Cat No. | Species | Antibody Name | Format | Classified by tag | Detail |
|---|
| GM-Tg-hg-T99816-Ab | Human | Anti-Human GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-rg-T99816-Ab | Rat | Anti-Rat GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-mg-T99816-Ab | Mouse | Anti-Mouse GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-cynog-T99816-Ab | Cynomolgus/Rhesus macaque | Anti-Cynomolgus/Rhesus macaque GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-felg-T99816-Ab | Cat/Feline | Anti-Cat/Feline GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-cang-T99816-Ab | Dog/Canine | Anti-Dog/Canine GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-bovg-T99816-Ab | Bovines/Cattle | Anti-Bovines/Cattle GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-equg-T99816-Ab | Equine/Horse | Anti-Equine/Horse GRPR monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
GRPR VLP (virus-like particle)/protein
| Cat No. | Species | Antigen Name | Expression Platform | Detail |
|---|
| GM-Tg-hg-T99816-Ag | Human | Human GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-rg-T99816-Ag | Rat | Rat GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-mg-T99816-Ag | Mouse | Mouse GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-cynog-T99816-Ag | Cynomolgus/Rhesus macaque | Cynomolgus/Rhesus macaque GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-felg-T99816-Ag | Cat/Feline | Cat/Feline GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-cang-T99816-Ag | Dog/Canine | Dog/Canine GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-bovg-T99816-Ag | Bovines/Cattle | Bovines/Cattle GRPR VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-equg-T99816-Ag | Equine/Horse | Equine/Horse GRPR VLP (virus-like particle) | HEK293 | Products Developing |