GRPR Target & Gene Products-cDNA ORF clones/siRNA/antibody/protein

Explore GRPR gene products and cross-species research data at TarMart platform. Discover comprehensive biological information, expression tools, and therapeutic insights for Homo sapiens (human), Cynomolgus monkeys, rodents (mouse/rat), canines, felines, bovines, and equines. Your premier destination for multi-species gene research solutions
Target sublocation: Transmembrane Protein.
Gastrin-releasing peptide (GRP) regulates numerous functions of the gastrointestinal and central nervous systems, including release of gastrointestinal hormones, smooth muscle cell contraction, and epithelial cell proliferation and is a potent mitogen for neoplastic tissues. The effects of GRP are mediated through the gastrin-releasing peptide receptor. This receptor is a glycosylated, 7-transmembrane G-protein coupled receptor that activates the phospholipase C signaling pathway. The receptor is aberrantly expressed in numerous cancers such as those of the lung, colon, and prostate. An individual with autism and multiple exostoses was found to have a balanced translocation between chromosome 8 and a chromosome X breakpoint located within the gastrin-releasing peptide receptor gene. [provided by RefSeq, Jul 2008]

Target ID GM-T99816
Target Name GRPR
Gene Group ldentifer
(Target Gene ID in Homo species)
2925
Gene ID 100056400 (Equus caballus), 101096951 (Felis catus), 14829 (Mus musculus), 24938 (Rattus norvegicus)
2925 (Homo sapiens), 491754 (Canis lupus familiaris), 532784 (Bos taurus), 574339 (Macaca mulatta)
Target Alternative Names BB2,BB2R,BRS2,GRP-R,GRP-preferring bombesin receptor,GRPR,Gastrin-releasing peptide receptor,Grpr
Uniprot Accession P21729,P52500,P30550
Protein Sub-location Transmembrane Protein
Category Therapeutics Target
Disease from KEGG Calcium signaling pathway, Neuroactive ligand-receptor interaction
Gene Ensembl ENSECAG00000015277, ENSMUSG00000031364, ENSG00000126010, ENSCAFG00845030779, ENSBTAG00000007092, ENSMMUG00000023688
Target Classification GPCR


Pre-made viral vector of GRPR cDNA Clones/ORF Plasmid

Cat No.Product NameNMIDGeneIDSpeciesTypeMarkerFusion TagPromoterDetail
pGMLP003622Human GRPR/BB2/BB2R Lentivirus plasmidNM_0053142925HumanLentivirus plasmidZsGreen3xflag (C-Terminal)CMVDetail
pGMPC000580Human GRPR/BB2/BB2R Mammalian (Non-Viral Vector) plasmidNM_005314.32925HumanMammalian (Non-Viral Vector) plasmidNull3xflag (C-Terminal)CMVDetail
pGMPC000624Human GRPR/BB2/BB2R Mammalian (Non-Viral Vector) plasmidNM_005314.32925HumanMammalian (Non-Viral Vector) plasmidEGFP3xflag (C-Terminal)EF1Detail
vGMLP003622Human GRPR/BB2/BB2R Lentivirus particleNM_0053142925HumanLentivirus particleZsGreen3xflag (C-Terminal)CMVDetail
pGMAAV001593Mouse Grpr/GRP-R Adeno-associate virus(AAV) plasmidNM_00817714829MouseAdeno-associate virus(AAV) plasmidNull3xflag (C-Terminal)F4/80Detail
pGMLPm002318Mouse Grpr/GRP-R Lentivirus plasmidNM_00817714829MouseLentivirus plasmidZsGreen3xflag (C-Terminal)CMVDetail
pGMPC000238Mouse GRPR/GRP-R Mammalian (Non-Viral Vector) plasmidNM_00817714829MouseMammalian (Non-Viral Vector) plasmidZsGreen3xflag (C-Terminal)CMVDetail
vGMAAV001593Mouse Grpr/GRP-R Adeno-associate virus(AAV) particleNM_00817714829MouseAdeno-associate virus(AAV) particleNull3xflag (C-Terminal)F4/80Detail
vGMLPm002318Mouse Grpr/GRP-R Lentivirus particleNM_00817714829MouseLentivirus particleZsGreen3xflag (C-Terminal)CMVDetail


GRPR siRNA/miRNA/oligo for RNA interfence (RNAi)

Cat No.Product NameGeneIDSpeciesGradeDetail
pGMoligo2925Pre-made Human GRPR/BB2/BB2R siRNA oligo Duplex2925HumanIn-vitro grade; in-vivo gradeDetail
pGMoligo24938Pre-made Rat Grpr siRNA oligo Duplex24938RatIn-vitro grade; in-vivo gradeDetail
pGMoligo14829Pre-made Mouse Grpr/GRP-R siRNA oligo Duplex14829MouseIn-vitro grade; in-vivo gradeDetail
pGMoligo574339Pre-made Cynomolgus/Rhesus macaque GRPR siRNA oligo Duplex574339Cynomolgus/Rhesus macaqueIn-vitro grade; in-vivo gradeDetail
pGMoligo101096951Pre-made Cat/Feline GRPR siRNA oligo Duplex101096951Cat/FelineIn-vitro grade; in-vivo gradeDetail
pGMoligo491754Pre-made Dog/Canine GRPR siRNA oligo Duplex491754Dog/CanineIn-vitro grade; in-vivo gradeDetail
pGMoligo532784Pre-made Bovines/Cattle GRPR siRNA oligo Duplex532784Bovines/CattleIn-vitro grade; in-vivo gradeDetail
pGMoligo100056400Pre-made Equine/Horse GRPR siRNA oligo Duplex100056400Equine/HorseIn-vitro grade; in-vivo gradeDetail


GRPR antibody/GMab

Cat No.SpeciesAntibody NameFormatClassified by tagDetail
GM-Tg-hg-T99816-AbHumanAnti-Human GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-rg-T99816-AbRatAnti-Rat GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-mg-T99816-AbMouseAnti-Mouse GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-cynog-T99816-AbCynomolgus/Rhesus macaqueAnti-Cynomolgus/Rhesus macaque GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-felg-T99816-AbCat/FelineAnti-Cat/Feline GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-cang-T99816-AbDog/CanineAnti-Dog/Canine GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-bovg-T99816-AbBovines/CattleAnti-Bovines/Cattle GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail
GM-Tg-equg-T99816-AbEquine/HorseAnti-Equine/Horse GRPR monoclonal antibodymabFACS/Biofunctional Antibody, Therapeutics Target antibodyDetail


GRPR VLP (virus-like particle)/protein

Cat No.SpeciesAntigen NameExpression PlatformDetail
GM-Tg-hg-T99816-AgHumanHuman GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-rg-T99816-AgRatRat GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-mg-T99816-AgMouseMouse GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-cynog-T99816-AgCynomolgus/Rhesus macaqueCynomolgus/Rhesus macaque GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-felg-T99816-AgCat/FelineCat/Feline GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-cang-T99816-AgDog/CanineDog/Canine GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-bovg-T99816-AgBovines/CattleBovines/Cattle GRPR VLP (virus-like particle)HEK293Products Developing
GM-Tg-equg-T99816-AgEquine/HorseEquine/Horse GRPR VLP (virus-like particle)HEK293Products Developing