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Target
sublocation: Transmembrane Protein.
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors H1, H2, H3 and H4. The protein encoded by this gene is an integral membrane protein and belongs to the G protein-coupled receptor superfamily. It mediates the contraction of smooth muscles, the increase in capillary permeability due to contraction of terminal venules, the release of catecholamine from adrenal medulla, and neurotransmission in the central nervous system. It has been associated with multiple processes, including memory and learning, circadian rhythm, and thermoregulation. It is also known to contribute to the pathophysiology of allergic diseases such as atopic dermatitis, asthma, anaphylaxis and allergic rhinitis. Multiple alternatively spliced variants, encoding the same protein, have been identified. [provided by RefSeq, Jan 2015]
| Target ID |
GM-T77913
|
| Target Name |
HRH1/H1R
|
Gene Group ldentifer (Target Gene ID in Homo
species)
|
3269
|
| Gene ID |
100034110 (Equus caballus), 101088314 (Felis catus), 15465 (Mus musculus), 24448 (Rattus norvegicus) 281231 (Bos taurus), 3269 (Homo sapiens), 403813 (Canis lupus familiaris), 696359 (Macaca mulatta)
|
| Target Alternative Names |
Bphs,H1,H1-R,H1R,HH1R,HRH1,Hir,Hisr,Histamine H1 receptor,Hrh1,hisH1
|
| Uniprot Accession |
P70174,P31390,P30546,P35367
|
| Protein Sub-location |
Transmembrane Protein
|
| Category |
Therapeutics Target
|
| Disease from KEGG |
Calcium signaling pathway, Neuroactive ligand-receptor interaction, Inflammatory mediator regulation of TRP channels
|
| Gene Ensembl |
ENSECAG00000004544, ENSMUSG00000053004, ENSBTAG00000061643, ENSG00000196639, ENSCAFG00845006605, ENSMMUG00000056308
|
| Target Classification |
GPCR
|
Pre-made viral vector of HRH1/H1R cDNA Clones/ORF Plasmid
HRH1/H1R siRNA/miRNA/oligo for RNA interfence (RNAi)
| Cat No. | Product Name | GeneID | Species | Grade | Detail |
|---|
| pGMoligo3269 | Pre-made Human HRH1/H1R/H1-R siRNA oligo Duplex | 3269 | Human | In-vitro grade; in-vivo grade | Detail |
| pGMoligo24448 | Pre-made Rat Hrh1/Hisr siRNA oligo Duplex | 24448 | Rat | In-vitro grade; in-vivo grade | Detail |
| pGMoligo15465 | Pre-made Mouse Hrh1/H1R/Hir siRNA oligo Duplex | 15465 | Mouse | In-vitro grade; in-vivo grade | Detail |
| pGMoligo696359 | Pre-made Cynomolgus/Rhesus macaque HRH1 siRNA oligo Duplex | 696359 | Cynomolgus/Rhesus macaque | In-vitro grade; in-vivo grade | Detail |
| pGMoligo101088314 | Pre-made Cat/Feline HRH1 siRNA oligo Duplex | 101088314 | Cat/Feline | In-vitro grade; in-vivo grade | Detail |
| pGMoligo403813 | Pre-made Dog/Canine HRH1 siRNA oligo Duplex | 403813 | Dog/Canine | In-vitro grade; in-vivo grade | Detail |
| pGMoligo281231 | Pre-made Bovines/Cattle HRH1 siRNA oligo Duplex | 281231 | Bovines/Cattle | In-vitro grade; in-vivo grade | Detail |
| pGMoligo100034110 | Pre-made Equine/Horse HRH1/H1 siRNA oligo Duplex | 100034110 | Equine/Horse | In-vitro grade; in-vivo grade | Detail |
HRH1/H1R antibody/GMab
| Cat No. | Species | Antibody Name | Format | Classified by tag | Detail |
|---|
| GM-Tg-hg-T77913-Ab | Human | Anti-Human HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-rg-T77913-Ab | Rat | Anti-Rat HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-mg-T77913-Ab | Mouse | Anti-Mouse HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-cynog-T77913-Ab | Cynomolgus/Rhesus macaque | Anti-Cynomolgus/Rhesus macaque HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-felg-T77913-Ab | Cat/Feline | Anti-Cat/Feline HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-cang-T77913-Ab | Dog/Canine | Anti-Dog/Canine HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-bovg-T77913-Ab | Bovines/Cattle | Anti-Bovines/Cattle HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
| GM-Tg-equg-T77913-Ab | Equine/Horse | Anti-Equine/Horse HRH1/H1R monoclonal antibody | mab | FACS/Biofunctional Antibody, Therapeutics Target antibody | Detail |
HRH1/H1R VLP (virus-like particle)/protein
| Cat No. | Species | Antigen Name | Expression Platform | Detail |
|---|
| GM-Tg-hg-T77913-Ag | Human | Human HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-rg-T77913-Ag | Rat | Rat HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-mg-T77913-Ag | Mouse | Mouse HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-cynog-T77913-Ag | Cynomolgus/Rhesus macaque | Cynomolgus/Rhesus macaque HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-felg-T77913-Ag | Cat/Feline | Cat/Feline HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-cang-T77913-Ag | Dog/Canine | Dog/Canine HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-bovg-T77913-Ag | Bovines/Cattle | Bovines/Cattle HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |
| GM-Tg-equg-T77913-Ag | Equine/Horse | Equine/Horse HRH1/H1R VLP (virus-like particle) | HEK293 | Products Developing |